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Brain Health Pikamilone Nootropics Powder

Brain Health Pikamilone Nootropics Powder

Brain Health Pikamilone Nootropics Powder Pikamilone Quick Detail: Product Name: Pikamilone Synonyms: PIKAMILONE HYDROCHLORIDE;NICOTINOYL-GABA;N-(3-CARBOXYPROPYL) NICOTINAMIDE;4-[(PYRIDIN-3-YLCARBONYL)AMINO]BUTANOIC ACID;4-(NICOTINAMIDO)BUTANOIC ACID;4-(3-PYRIDYLCARBOXAMIDO)BUTYRIC...

Product Details

Brain Health Pikamilone Nootropics Powder

Pikamilone Quick Detail:

Product Name: Pikamilone
Synonyms: PIKAMILONE HYDROCHLORIDE;NICOTINOYL-GABA;N-(3-CARBOXYPROPYL) NICOTINAMIDE;4-[(PYRIDIN-3-YLCARBONYL)AMINO]BUTANOIC ACID;4-(NICOTINAMIDO)BUTANOIC ACID;4-(3-PYRIDYLCARBOXAMIDO)BUTYRIC ACID;4-[(3-PYRIDINYLCARBONYL)AMINO]BUTANOIC ACID;Pikamiline
CAS: 34562-97-5
MF: C10H12N2O3
MW: 208.21
Product Categories: Heterocycles;Chemistry;API;Other APIs
Appearance Crystal powder
Application Smart nutrition

Pikamilone Description

Picamilon is a dietary supplement and nootropic drug. It is a combination of Vitamin B3, also known as niacin, and the neurotransmitter GABA. This supplement is taken orally, typically in powder or tablet form, and is able to cross the blood-brain barrier. Once in the brain, it is hydrolyzed into GABA and niacin.


The function of picamilon is two-fold, since, when the compound is broken down into its constituent parts in the brain, each one has a different effect. Niacin acts as a vasodilator, which enlarges the blood vessels of the brain. This, in turn, leads to increased blood flow, reduced blood pressure, and is thought to assist in the management of migraine headache pain.


When the second part of the picamilon compound, GABA, is activated in the brain, it is a believed to create a moderate anti-anxiety effect. This is known as an anxiolytic response, and is due to that fact that GABA is an inhibitory neurotransmitter. GABA limits, rather than encourages, certain brain functions.

Pikamilone Usage

The primary Nootropic benefits of Picamilon center on mood boosting and overall brain function improvements. This includes helping toreduce feelingsof stress and anxiety.


In fact, many users feel that Picamilon is so good at reducing these feelings that they use Picamilon on a regular basis to help relax. An improved positive outlook and attitude will also often follow. Once a person is relaxed, they will usually find themselves having improved sleep which is also more restful and deeper.

As a brain booster, Picamilon benefits also include better mental energy and improved clarity and focus. It is easier to think and make decisions as well when using Picamilon supplements.


There are also a number of additional health benefits associated with daily dosages of Picamilon nootropic. For starters, Picamilon helps to reduce and regulate blood pressure in the body. There is also a lot of evidence demonstrating that it can alleviate migraines and poor cerebral blood flow and circulation.


This supplement has further been shown to treat the symptoms of acute alcohol intoxication and the effects upon the brain. There is even the possibility that Picamilon may act as an anti-oxidant and rid the brain of toxins and other harmful substances.


Pikamilone Application

It is helpful to think of Picamilon as a mixture of two different chemicals – GABA and Niacin.

Once it is absorbed into the bloodstream both compounds cross over the blood-brain barrier together. This is courtesy of the Niacin pathways since GABA is not capable of this action by itself.


As the GABA enters into the central nervous system it targets receptor sites and performs its job as the chief inhibitory neurotransmitter within the human body. GABA is known to prevent over-stimulation and excitotoxicity of your brain cells which can occur when your neurons are firing faster than they should be.

We experience this over-activity as anxiety and the feeling like you cannot stop thinking about certain memories or future possibilities. Picamilon essentially curbs these excessive thought processes, resulting in a sensation of peace and calm.


Many people are tempted to think of the Niacin found in Picamilon powder simply as a GABA transport method. They would be incorrect; the Niacin from Picamilon is itself active and has a positive nootropic effect on mental performance. This substance is primarily responsible for opening up (or dilating) blood vessels within the brain.


As these passageways open, this leads to the improvement in cerebral blood flow, oxygen supply and glucose metabolism. The result is better cellular energy and improved resource supply to maintain the health of your neurons.


It also helps to keep skin healthy and may even play a role in improving vision in those suffering from glaucoma.


Pikamilone Dosage


The standard dosage range for Picamilon is between 50 and 300 mg per day.Of course, this may be split into several different administrations throughout the day, depending upon how it effects the user. Generally, a divided dose means one in the morning and one in the evening.


Most supplements sell it in 150 mg tablets or capsules, but you can also buy it as a bulk powder to get more control over your dosages. Picamilon works best when taken on an empty stomach and the effects of this nootropic will last anywhere from two to four hours.


You should always start out with the smallest effective Picamilon dose possible. Study the benefits obtained and then determine if increasing the dose is in order.


Pikamilone Stacking & Cycling Picamilon


Many users have found that stacking and cycling their Picamilon dosages can be very effective. It is certainly very safe and it may even help to increase the effects of other Nootropic supplements like the Racetams including Aniracetam and Piracetam. Even herbs like Valerian Root and Kava can be helpful when used in combination.


There are a number of other Nootropics that have similar effects to Picamilon, but might lead to tolerance if used on a daily basis. This means that it might be helpful to include Picamilon as part of a cycle with something like, say, Phenibut.


Start with the safer option (Picamilon) and use on a 3 or 4 day on and 2 day off cycle. For the days off of Picamilon, substitute with the Phenibut.


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